| 1. Hertzel AV, Hellberg K, Reynolds JM, Kruse AC, Juhlmann BE, Smith AJ, Sanders MA, Ohlendorf DH, Suttles J, Bernlohr DA. (2009) Identification and characterization of a small molecule inhibitor of Fatty Acid binding proteins.. J Med Chem, 52 (19): (6024-31). [PMID:19754198] [10.1021/op500134e] |
| 2. Liu X, Huang X, Lin W, Wang D, Diao Y, Li H, Hui X, Wang Y, Xu A, Wu D et al.. (2011) New aromatic substituted pyrazoles as selective inhibitors of human adipocyte fatty acid-binding protein.. Bioorg Med Chem Lett, 21 (10): (2949-52). [PMID:21481589] [10.1021/op500134e] |
| 3. Oddi S, Scipioni L, Totaro A, Angelucci C, Dufrusine B, Sabatucci A, Tortolani D, Coletta I, Alisi MA, Polenzani L et al.. (2019) The anti-inflammatory agent bindarit acts as a modulator of fatty acid-binding protein 4 in human monocytic cells.. Sci Rep, 9 (1): (15155). [PMID:31641194] [10.1021/op500134e] |
| 4. Haiyan Cai,Guirui Yan,Xiaodong Zhang,Olena Gorbenko,Heyao Wang,Weiliang Zhu. (2010-05-18) Discovery of highly selective inhibitors of human fatty acid binding protein 4 (FABP4) by virtual screening.. Bioorganic & medicinal chemistry letters, 20 ((12)): (3675-3679). [PMID:20471252] |
| 5. Lehmann F, Haile S, Axen E, Medina C, Uppenberg J, Svensson S, Lundbäck T, Rondahl L, Barf T.. (2004) Discovery of inhibitors of human adipocyte fatty acid-binding protein, a potential type 2 diabetes target.. Bioorg Med Chem Lett, 14 (17): (4445-4448). [PMID:15357969] [10.1016/j.bmcl.2004.06.057] |
| 6. Barf T, Lehmann F, Hammer K, Haile S, Axen E, Medina C, Uppenberg J, Svensson S, Rondahl L, Lundbäck T.. (2009) N-Benzyl-indolo carboxylic acids: Design and synthesis of potent and selective adipocyte fatty-acid binding protein (A-FABP) inhibitors.. Bioorg Med Chem Lett, 19 (6): (1745-1748). [PMID:19217286] [10.1016/j.bmcl.2009.01.084] |
| 7. Cai H, Liu Q, Gao D, Wang T, Chen T, Yan G, Chen K, Xu Y, Wang H, Li Y, Zhu W.. (2015) Novel fatty acid binding protein 4 (FABP4) inhibitors: virtual screening, synthesis and crystal structure determination.. Eur J Med Chem, 90 (241-250). [PMID:25461324] [10.1016/j.ejmech.2014.11.020] |
| 8. Zhou Y, Nie T, Zhang Y, Song M, Li K, Ding M, Ding K, Wu D, Xu Y.. (2016) The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation.. Bioorg Med Chem, 24 (18): (4310-4317). [PMID:27460668] [10.1016/j.bmc.2016.07.022] |
| 9. Kühne H, Obst-Sander U, Kuhn B, Conte A, Ceccarelli SM, Neidhart W, Rudolph MG, Ottaviani G, Gasser R, So SS, Li S, Zhang X, Gao L, Myers M.. (2016) Design and synthesis of selective, dual fatty acid binding protein 4 and 5 inhibitors.. Bioorg Med Chem Lett, 26 (20): (5092-5097). [PMID:27658368] [10.1016/j.bmcl.2016.08.071] |
| 10. Gao DD, Dou HX, Su HX, Zhang MM, Wang T, Liu QF, Cai HY, Ding HP, Yang Z, Zhu WL, Xu YC, Wang HY, Li YX.. (2018) From hit to lead: Structure-based discovery of naphthalene-1-sulfonamide derivatives as potent and selective inhibitors of fatty acid binding protein 4.. Eur J Med Chem, 154 (44-59). [PMID:29775936] [10.1016/j.ejmech.2018.05.007] |
| 11. Yan S, Elmes MW, Tong S, Hu K, Awwa M, Teng GYH, Jing Y, Freitag M, Gan Q, Clement T, Wei L, Sweeney JM, Joseph OM, Che J, Carbonetti GS, Wang L, Bogdan DM, Falcone J, Smietalo N, Zhou Y, Ralph B, Hsu HC, Li H, Rizzo RC, Deutsch DG, Kaczocha M, Ojima I.. (2018) SAR studies on truxillic acid mono esters as a new class of antinociceptive agents targeting fatty acid binding proteins.. Eur J Med Chem, 154 (233-252). [PMID:29803996] [10.1016/j.ejmech.2018.04.050] |
| 12. He Y, Dou H, Gao D, Wang T, Zhang M, Wang H, Li Y.. (2019) Identification of new dual FABP4/5 inhibitors based on a naphthalene-1-sulfonamide FABP4 inhibitor.. Bioorg Med Chem, 27 (19): (115015-115015). [PMID:31420256] [10.1016/j.bmc.2019.07.031] |
| 13. Oukoloff K, Lucero B, Francisco KR, Brunden KR, Ballatore C.. (2019) 1,2,4-Triazolo[1,5-a]pyrimidines in drug design.. Eur J Med Chem, 165 (332-346). [PMID:30703745] [10.1016/j.ejmech.2019.01.027] |
| 14. Baxa, C A CA and 7 more authors.. (1989) Human adipocyte lipid-binding protein: purification of the protein and cloning of its complementary DNA.. Biochemistry, (31): [PMID:2481498] |
| 15. Bienvenut, Willy V WV and 6 more authors.. (2012) Comparative large scale characterization of plant versus mammal proteins reveals similar and idiosyncratic N-α-acetylation features.. Molecular & cellular proteomics : MCP, [PMID:22223895] |
| 16. Rosenow, Anja A and 6 more authors.. (2012) Resveratrol-induced changes of the human adipocyte secretion profile.. Journal of proteome research, (7): [PMID:22905912] |
ZJ23F0800875